%0 Journal Article %K molecular dynamics %K Calorimetry %K selective inhibitors %K Crystallography %K X-Ray %K BRPF1 %B European Journal of Medicinal Chemistry %D 2018 %G eng %N 155 %P 337-352 %R 10.1016/j.ejmech.2018.05.037 %T Structure-based discovery of selective BRPF1 bromodomain inhibitors %U https://www.sciencedirect.com/science/article/pii/S0223523418304501 %1 0236 %8 May 23 2018 %9 Research Article %& 337